GRK3

G protein-coupled receptor kinase 3 P35626 GRK3_HUMAN
Protein Coding Chr 22 22q12.1 Swiss-Prot reviewed Entrez 157
Mutations
304
CL 58 · Tissue 242
Samples
296
CL 57 · Tissue 236
Peptides
223
unique mutant peptides
Transcripts
1
isoforms mutated

Stats by Source

Total, split by cell line (COSMIC CL / DepMap / PubMed) vs tissue (COSMIC primary tissue)

How the counts split by source
Stats by Source

Total = all mutations for this gene across every source.

Cell line = COSMIC Cell Lines Project + DepMap + PubMed.

Tissue = COSMIC primary-tissue (patient tumour) samples.

Total can exceed cell line + tissue: COSMIC tissue-derived models sit only in global, and a peptide can be shared across both.

TotalCell lineTissue
Mutations30458242
Samples29657236
Peptides22340186

Function

GRK3 · G protein-coupled receptor kinase 3

The beta-adrenergic receptor kinase specifically phosphorylates the agonist-occupied form of the beta-adrenergic and related G protein-coupled receptors. Overall, the beta adrenergic receptor kinase 2 has 85% amino acid similarity with beta adrenergic receptor kinase 1, with the protein kinase catalytic domain having 95% similarity. These data suggest the existence of a family of receptor kinases which may serve broadly to regulate receptor function. [provided by RefSeq, Jul 2008].

Isoforms & Proteins

1 transcript · UniProt mapping is sequence-verified (AA-safe)

About the isoform mapping
Isoforms & Proteins

Each Ensembl transcript (ENST) this gene is mutated on, with its matched UniProt accession.

The mapping is sequence-verified: the UniProt sequence is identical to the transcript translation, so amino-acid positions line up exactly. A * marks an unreviewed (TrEMBL) entry.

Counts are mutations and unique mutant peptides on each transcript.

TranscriptUniProtMutationsPeptides
ENST00000324198 P35626 304 223

Gene Properties

Type
Protein Coding
Chromosome
22
Cytoband
22q12.1
Entrez ID
Aliases
ADRBK2BARK2

Recurrent Mutations

All 223 amino-acid changes on canonical ENST00000324198 · needle height = samples · drag the mini-map to zoom

What this lollipop shows
Recurrent Mutations

A lollipop / needle plot – the standard way to show recurrent mutations along a protein (as used by cBioPortal and MutationMapper).

X-axis = amino-acid position in the protein.

Needle height & head size = how often that exact amino-acid change was observed (its recurrence). Tall/large heads are mutational hotspots.

The most recurrent changes are labelled; hover any needle for the change, position and counts.

Mutation frequency across cancer types

% of samples with a missense/complex mutation in GRK3 · cell line vs tissue

How this frequency is counted
Cancer-type mutation frequency

For each cancer type, the fraction of samples that carry at least one missense/complex mutation anywhere in GRK3 – counted as distinct samples (a sample counts once no matter how many mutations it has).

Split into cell line and tissue; each cell shows mutated / total and the percentage. Cohorts with <20 samples are omitted. Ordered by combined frequency.

Cancer typeCell linesTissue samples
Oral Cavity Carcinoma
5/54 9%
0/0 0%
T-Lymphoblastic Leukemia
2/40 5%
0/0 0%
T-Cell Non-Hodgkins Lymphoma
1/26 4%
0/0 0%
Endometrial Carcinoma
5/42 12%
20/612 3%
Other Solid Cancers
0/94 0%
23/1515 2%
Colorectal Carcinoma
12/143 8%
35/3239 1%
Melanoma
4/210 2%
25/1899 1%
Small Cell Lung Carcinoma
0/9 0%
9/752 1%
Neuroendocrine Tumour
6/154 4%
2/577 0%
Cervical Carcinoma
0/35 0%
5/422 1%
Gastric Carcinoma
1/74 1%
16/1809 1%
Ovarian Carcinoma
4/109 4%
6/998 1%
Burkitts Lymphoma
0/32 0%
2/196 1%
Non-Small Cell Lung Carcinoma
2/304 1%
10/1390 1%
Other Sarcomas
1/69 1%
4/699 1%
Glioma
2/52 4%
10/2127 0%
Non-Cancerous
0/104 0%
5/830 1%
Germ Cell Tumour
0/25 0%
1/169 1%
Hepatocellular Carcinoma
0/46 0%
11/2210 0%
Bladder Carcinoma
3/58 5%
2/956 0%
Osteosarcoma
1/45 2%
0/166 0%
Mesothelioma
0/62 0%
1/165 1%
Biliary Tract Carcinoma
0/54 0%
4/950 0%
Kidney Carcinoma
0/85 0%
7/1862 0%
B-Cell Non-Hodgkins Lymphoma
1/88 1%
8/2534 0%
Thyroid Gland Carcinoma
0/45 0%
5/1592 0%
Esophageal Squamous Cell Carcinoma
0/51 0%
8/2550 0%
Plasma Cell Myeloma
0/44 0%
1/305 0%
Breast Carcinoma
0/144 0%
9/3264 0%
Head and Neck Carcinoma
0/85 0%
4/1574 0%

Mutation Distribution

Where GRK3 is mutated · all tissues, split by cell line vs tissue

Mutation counts by tissue
Mutation Distribution

How many mutations in GRK3 were found in each tissue, across the whole database.

Each bar is a tissue (cell-line and tissue names are merged to the standard tissue), split into cell line and tissue (patient tumour) contributions.

This shows the cancer-context where this gene is recurrently altered.

GTEx Expression

Median TPM across 54 healthy tissues

GTEx Portal ↗
About the expression data
GTEx Expression

Median gene expression (TPM) in normal, non-cancer human tissues from the GTEx project.

Useful for judging tumour specificity – a strong neoantigen target ideally comes from a gene with low expression in healthy tissues.

Scroll or drag the mini-axis below the chart to browse all tissues.

Mutations

All 304 mutations in GRK3

About the mutation list
Mutations

Every mutation record for this gene, across all samples and sources.

The Sample column links to the cell line (cell-line samples) or the tissue type (tissue samples).

Use the Type / Source filters, the search box, and column sorting to explore; each CAN-IMMUNE ID opens the full mutation & peptide view.

IDSampleTranscriptAA Change CDSTypeSourceMutant PeptideWild-type Peptide